Ac-Lys-Val-Cit-PABC-MMAE formic
| Specifications | |
|---|---|
| Formula: | C67H110N12O16 |
| Molecular Weight: | 1339,66 |
Description
Ac-Lys-Val-Cit-PABC-MMAE (formic) is an agent-linker conjugate utilized in antibody-drug conjugates (ADCs). This compound comprises a peptide linker (Ac-Lys-Val-Cit-PABC) attached to the cytotoxic agent Monomethyl auristatin E (MMAE), which serves as a potent inhibitor of tubulin polymerization[1].
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